A spoiled rich kid from Hong Kong, Huang Lee owes his status as a Triad member to his father, a Triad boss from Kowloon. After the murder of his father, Huang is called to Liberty City by his Uncle Wu "Kenny" Lee to deliver a family 'heirloom", the Yu Jian Sword, to secure his family's claim to the leadership of the Triad gangs. But what was supposed to be a weekend of table service and strippers turns into a dangerous adventure after arriving at Francis International Airport only to be hijacked, robbed of his sword, and left for dead. Huang will have to dig deep into the rotten core of Liberty City - and deep within himself -- to avenge his father's murder and reclaim his family's honor.
The leader of the Lee Clan within the Triad organizations of Liberty City, Uncle Kenny is from the old school. He likes his suits double breasted, his platitudes from a fortune cookie, and his payments in cash. Uncle Kenny wants control of the Triads, and there is little that he won't ask Huang to do for him to get it.
A dirty narcotics detective with the IAD on his tail and a monkey on his back, Wade Heston forms a dubious alliance with Huang Lee to find the mysterious FIB rat who has set up both Huang and Wade. Lying, stealing and murdering are all in a day’s work for this member of Liberty City’s finest.
Hsin Jaoming has ruled the Triad gangs of Liberty City for over twenty years with an iron fist. But now nearing retirement, he is looking for a worthy successor with as much ambition and brains as himself.
The son of Liberty City Triad boss Hsin Jaoming, Chan is a willful, drug-addled and stupid playboy. Chan buys his friends and makes his enemies with little caution and even less thought.
Zhou Ming is the leader of the Ming Family and might be another rival of Huang Lee and the Lee Family.
Lester Leroc is a private investigator who is working for Hsin Jaoming. He is undercover with the Angels of Death to find out if there is a rat in the Angels. He asks Huang to help him out with some things he can't do himself.
Rudy D'Avanzo is an Italian gangster. He contacts Huang, saying he knows who the rat is. He tells that it's name is Jimmy Capra. Rudy asks Huang to do some things for him in exchange for a tape with evidence Jimmy is the rat.
Xin Shan is a Chinese ganster. After you found the two Lions of Fo, you are able to download his missions at the Rockstar Social Club. He asks you to help him out with some things, because his partner was killed. He is the brother of Ling Shan.
Ling Shan is a street smart Chinatown girl whose beauty belies her deadly skills. She serves as Uncle Kenny's master at arms, and provides necessary muscle in a town that only respects money and brute force. Trained in the martial arts and deadly with all manner of small arms, it is Ling who teaches Huang the combat skills he will need to survive on the streets of Liberty City.
Jimmy Capra is the fed rat, according to Rudy D'Avanzo. He meets with Rudy for a 'peace talk', but it doesn't end well for him.